Endocrinology — Drugs

(products approved for use in Canada)

Drug Class

Generic Name(s)

Trade Name(s)

Growth Hormones

somatropin

Humatrope, Nutropin, Saizen

Somatostatin Analogues

octreotide

Sandostatin, Sandostatin LAR

somatostatin

Stilamin

Posterior Pituitary Hormones

desmopressin

DDAVP, Minirin, Octostim

vasopressin (ADH)

Pressyn

Dopamine Agonists

bromocriptine

Parlodel

cabergoline

Dostinex

quinagolide

Norprolac

Thyroid Hormones

levothyroxine sodium

Eltroxin, Synthroid

liothyronine sodium

Cytomel

thyroid, dessicated

Thyroid

Thyrotropin Releasing Hormone (TRH)

protirelin

Relefact

Thyroid Stimulating Hormone (TSH)

thyrotropin alfa

Thyrogen

Iodides

potassium iodide

potassium iodide + iodine

Lugol’s Solution

Thioureylenes

methimazole

Tapazole

propylthiouracil (PTU)

Propyl-Thyracil

Parenteral Calcium

calcium gluconate

calcium chloride

Oral Calcium

calcium carbonate

Os-Cal, Calcite, Calsan, Caltrate

Calcimimetic

cinacalcet

Sensipar

Vitamin D and Analogues

alfacalcidol

One-Alpha

calcitriol

Rocaltrol, Calcijex

cholecalciferol (Vitamin D3)

dihydrotachysterol (DHT)

Hytakerol

ergocalciferol (Vitamin D2)

Drisdol, Ostoforte

Calcitonin

calcitonin salmon

Calcimar, Caltine, Miacalcin NS

Phosphate Binder

sevelamer

Renagel

Drug Class

Generic Name(s)

Trade Name(s)

Bisphosphonates

alendronate

Fosamax

clodronate

Bonefos, Ostac

etridronate

Didronel

ibandronate

Bondronat

pamidronate

Aredia

risedronate

Actonel

zoledronic acid

Zometa

Adrenocorticotropic Hormones

cosyntropin

Cortrosyn

Glucocorticoids

Oral

(Tablets, Liquid, Capsules)

betamethasone and sodium phosphate salt

Betnesol

budesonide

Entocort

cortisone acetate

Cortone

dexamethasone

hydrocortisone

Cortef

methylprednisolone

Medrol

prednisolone

Pediapred

prednisone

Winpred

Injectable

IV/IM

dexamethasone

Hexadrol

hydrocortisone sodium succinate

Solu-Cortef

methylprednisolone sodium succinate

Solu-Medrol

IM only

methylprednisolone acetate

Depo-Medrol

betamethasone sodium phosphate/acetate

Celestone Soluspan

triamcinolone acetonide

Kenalog

Intradermal

methylprednisolone acetate

Depo-Medrol

Drug Class

Generic Name(s)

Trade Name(s)

Glucocorticoids cont’d

Injectable cont’d

Intraarticular

betamethasone sodium phosphate/acetate

Celestone Soluspan

methylprednisolone acetate

Depo-Medrol

triamcinolone acetonide

Kenalog

triamcinolone hexacetonide

Aristospan

Inhalation

(Nasal, Pulmonary)

beclomethasone dipropionate

budesonide

Pulmicort, Rhinocort

flunisolide

Rhinalar

fluticasone

Flovent

triamcinolone acetonide

Azamacort, Nasacort

Ophthalmic

(Drops, Ointment)

betamethasone sodium phosphate

Betnesol

dexamethasone

Maxidex

fluorometholone

FML

hydrocortisone

prednisolone

Pred Forte, Pred Mild

rimexolone

Vexol

Otologic (ear)

betamethasone sodium phosphate

Betnesol

dexamethasone sodium

Rectal

(Enema, Foam, Ointment, Suppository)

betamethasone sodium phosphate

Betnesol

budesonide

Entocort

hydrocortisone and acetate salt

Cortenema, Cortifoam

Drug Class

Generic Name(s)

Trade Name(s)

 

Topical

(Cream, Lotion, Ointment)

amcinonide

Cyclocort

betamethasone benzoate, dipropionate, valerate

Betaderm, Betnovate, Celestoderm-V, Diprolone, Diprosone, Ectosone, Prevex B, Topilene, Topisone, Valisone

clobetasol propionate, butyrate

Dermasone, Dermovate, Eumovate

desonide

Desocort, Tridesilon

desoximetasone

Topicort

diflucortolone valerate

Merisone

fluocinolone acetonide

Derma-Smoothe FS, Fluoderm, Synalar

fluocinonide

Lidemol, Lidex, Lyderm, Lydonide, Tiamol, Topsyn

halcinonide

Halog

halobetasol

Ultravate

hydrocortisone

Aquacort, Cortate, Cortoderm, EmoCort, PrevexHC, Sarna HC

hydrocortisone acetate, valerate

Westcort

methylprednisolone, methylprednisolone acetate

Medrol

mometasone furoate

Elocom

triamcinolone acetonide

Aristocort, Kenalog, Triaderm

Mineralocorticoids

fludrocortisone acetate

Florinef

Insulins, Pork

insulin regular

insulin NPH

Insulins, Human

insulin regular

Humulin R, Novolin ge Toronto

insulin lente

Humulin L

insulin NPH

Humulin N, Novolin ge NPH

insulin ultralente

Humulin U

Drug Class

Generic Name(s)

Trade Name(s)

Insulins, Human, Mixed (Regular/NPH)

reg/NPH 10/90

Novolin ge 10/90

reg/NPH 20/80

Humulin 20/80, Novolin ge 20/80

reg/NPH 30/70

Humulin 30/70, Novolin ge 30/70

reg/NPH 40/60

Novolin ge 40/60

reg/NPH 50/50

Novolin ge 50/50

Insulin Analogues

insulin aspart

NovoRapid

insulin glargine

Lantus

insulin lispro

Humalog

insulin lispro 25% + neutral protamine lispro 75%

Humalog Mix 25

Sulfonylureas

chlorpropamide

gliclazide

Diamicron, Diamicron MR

glimepiride

Amaryl

glyburide

Diaβeta, Euglucon

tolbutamide

Meglitinides

nateglinide

Starlix

repaglinide

Gluconorm

Biguanide

metformin

Glucophage

α-Glucosidase Inhibitor

acarbose

Prandase

Thiazolidinediones (glitazones)

pioglitazone

Actos

rosiglitazone

Avandia

Combination Biguanide + Glitazone

metformin + rosiglitazone

Avandamet

Hyperglycemic Agents

diazoxide

Proglycem

glucagon

Phosphodiesterase (PDE-5) Inhibitors

sildenafil

Viagra

tadalafil

Cialis

vardenafil

Levitra

Oxytocic Agents

carbetocin

Duratocin

dinoprostone

Prostin E2 tablets, vaginal gel

ergonovine (ergometrine)

oxytocin

Drug Class

Generic Name(s)

Trade Name(s)

Estrogens

conjugated estrogens (oral,vaginal)

C.E.S., Congest, Premarin

dienestrol (vaginal)

Ortho-Dienestrol

esterified estrogens (oral, vaginal)

Neo-estrone

estradiol (oral)

Estrace

estradiol (transdermal)

Climara, Estraderm, Estrogel, Estradot, Oesclim, Rhoxal estradiol, Vivelle

estradiol (vaginal)

Estring, Vagifem

estradiol (injection)

Delestrogen, Neo-Diol

estrone (vaginal)

Neo-estrone vaginal cream

estropipate (oral)

Ogen

Progestins

medroxyprogesterone

Depo-Provera, Provera

megestrol

Megace

norethindrone

Micronor, Norlutate

progesterone, micronized

Prometrium, Crinone

Estrogen plus Progestin Combinations

estradiol + norethindrone

Estracomb, Estalis, Estalis Sequi

conjugated estrogens + medroxyprogesterone

Premplus

ethinyl estradiol + norethindrone

FemHRT

Estrogen plus Androgen

estradiol + testosterone

Climacteron

Estrogen plus Antiandrogen

ethinyl estradiol + cyproterone acetate

Diane-35

Selective Estrogen Receptor Modulators (SERMs)

raloxifene

Evista

Estrogen Agonist-Antagonists

clomiphene

Clomid

Hormonal Contraceptives

Transdermal

ethinyl estradiol / norelgestromin

Evra

Vaginal Ring

ethinyl estradiol / etonogestrel

NuvaRing

Drug Class

Generic Name(s)

Trade Name(s)

Hormonal Contraceptives cont’d

Monophasic

(< 50 mcg estrogen)

ethinyl estradiol / ethynodiol diacetate

Demulen 30

ethinyl estradiol / desogestrel

Marvelon, Ortho-Cept

ethinyl estradiol / drospirenone

Yasmin

ethinyl estradiol / levonorgestrel

Alesse, Min-Ovral

ethinyl estradiol / norethindrone

Brevicon 1/35, Ortho 0.5/35, Ortho 1/35, Select 1/35

ethinyl estradiol / norethindrone acetate

Minestrin 1/20, Loestrin 1.5/30

ethinyl estradiol / norgestimate

Cyclen

Monophasic

( 50 mcg estrogen)

ethinyl estradiol / ethynodiol diacetate

Demulen 50

ethinyl estradiol / norgestrel

Ovral

mestranol/ norethindrone

Norinyl 1/50, Ortho-Novum 1/50

Triphasic

ethinyl estradiol / levonorgestrel

Triphasil, Triquilar

ethinyl estradiol / norethindrone

Ortho 7/7/7, Synphasic

ethinyl estradiol / norgestimate

Tri-Cyclen, Tri-Cyclen Lo

Progestin Only

levonorgestrel

Mirena, Plan B

medroxyprogesterone

Depo-Provera

norethindrone

Micronor

Gonadotropin-Releasing Hormone (GnRH) Analogues

buserelin

Suprefact

gonadorelin

Lutrepulse

goserelin

Zoladex

leuprolide

Eligard, Lupron

nafarelin

Synarel

Drug Class

Generic Name(s)

Trade Name(s)

Gonadotropins

chorionic gonadotropin (human) (hCG)

Pregnyl

choriogonadotropin alfa

Ovidrel

follitropin alpha (FSH)

Gonal-F

follitropin beta (FSH)

Puregon

gonadotropin human (FSH and LH)

Humegon

menotropins (FSH and LH)

Pergonal

Gonadotropin-Releasing Hormone (GnRH) Antagonist

ganirelix

Orgalutran

Androgens

danazol

Cyclomen

fluoxymesterone

Halotestin

nandrolone decanoate

Deca-Durabolin

testosterone

Androderm, Androgel

testosterone cypionate

Depo-Testosterone

testosterone enanthate

Delatestryl

testosterone undecanoate

Andriol

Erectile Dysfunction Therapy

Oral Agents

sildenafil

Viagra

tadalafil

Cialis

vardenafil

Levitra

Intraurethral Agents

alprostadil

MUSE

Intracavernosal Injections

alprostadil

Caverject

papaverine

phentolamine

Regitine

Anorectics

diethylpropion

Tenuate, Tenuate Dospan

mazindol

Sanorex

phentermine

Ionamin

sibutramine

Meridia

Lipase Inhibitors

orlistat

Xenical






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