Gastrointestinal System – Drugs
(Products approved for use in Canada)
|
Drug Class |
Generic Name(s) |
Trade Name(s) |
|
Antacids |
aluminum hydroxide |
Amphojel |
|
aluminum hydroxide + magnesium hydroxide |
Diovol, Gelusil, Maalox |
|
calcium carbonate |
Tums |
|
calcium carbonate + magnesium hydroxide |
Rolaids |
|
magnesium hydroxide |
Phillips' Milk of Magnesia |
|
Antacid + Mucosal Anesthetic |
oxethazaine + aluminum and magnesium hydroxide |
Mucaine |
|
Alginate + Antacid |
alginic acid + aluminum hydroxide |
Gaviscon |
|
Prokinetic Agents |
domperidone |
|
|
erythromycin |
EES, Erybid, Eryc, Erythrocin |
|
metoclopramide |
|
|
H2 receptor Antagonists |
cimetidine |
|
|
famotidine |
Pepcid, Pepcid AC |
|
nizatidine |
Axid |
|
ranitidine |
Zantac |
|
Proton-Pump Inhibitors |
esomeprazole |
Nexium |
|
lansoprazole |
Prevacid |
|
omeprazole |
Losec |
|
pantoprazole |
Pantoloc, Panto IV |
|
rabeprazole |
Pariet |
|
Digestants (pancreatic enzymes) |
pancrelipase |
Cotazym, Creon, Pancrease, Ultrase, Viokase |
|
Litholytic Agents (gallstone dissolution) |
ursodeoxycholic acid or ursodiol |
Urso |
|
Drug Class |
Generic Name(s) |
Trade Name(s) |
|
Antiviral Agents for Chronic Hepatitis |
interferon alfa-2a |
Roferon-A |
|
interferon alfa-2b |
Intron A |
|
interferon alfacon-1 |
Infergen |
|
lamivudine |
Heptovir |
|
peginterferon alfa-2a |
Pegasys |
|
peginterferon alfa-2b |
Unitron PEG |
|
ribavirin + interferon alfa-2a |
Pegasys RBV |
|
ribavirin + interferon alfa-2b |
Rebetron |
|
ribavirin + peginterferon alfa-2b |
Pegetron |
|
Hepatitis Vaccines |
hepatitis A vaccine (inactivated) |
Avaxim, Epaxal, Havrix, Vaqta |
|
hepatitis B vaccine (recombinant) |
Energix-B, Recombivax HB |
|
hepatitis A & B vaccine |
Twinrix |
|
Cytoprotective Agents |
misoprostol |
|
|
sucralfate |
Sulcrate |
Laxatives |
|
|
|
Bulk-forming agents
|
methylcellulose |
Prodiem Bulk Fibre Therapy Powder |
|
polycarbophil calcium |
Prodiem Bulk Fibre Therapy Caplets |
|
psyllium |
Metamucil, Prodiem |
|
sterculia gum |
Normacol |
|
Stimulants
|
bisacodyl |
Carters Little Pills, Correctol, Dulcolax, Feen-A-Mint, |
|
cascara sagrada |
|
|
castor oil |
|
|
senna |
Ex-Lax, Nature’s Remedy, Prodiem Overnight Relief Therapy, Senokot |
|
Stool softeners |
docusate calcium or sodium |
Colace, Correctol Stool Softener |
|
Osmotic laxatives
|
glycerin |
Suppositories |
|
lactulose |
|
|
polyethylene glycol (PEG) + electrolytes |
Colyte, Klean-Prep, Lyteprep, PegLyte |
|
sorbitol |
|
|
Drug Class |
Generic Name(s) |
Trade Name(s) |
Laxatives |
|
|
|
Saline |
magnesium citrate |
Citro-Mag |
|
magnesium hydroxide |
Phillips Milk of Magnesia |
|
sodium phosphates |
Fleet Enema, Fleet Phosphosoda Oral Laxative, |
|
Lubricants
|
mineral oil |
Fleet Enema Mineral Oil, Lansoyl, Nujol, |
|
Antispasmodics |
|
|
|
Anticholinergics |
dicyclomine |
Bentylol |
|
glycopyrrolate |
|
|
hyoscine butylbromide |
Buscopan |
|
propantheline |
Propanthel |
|
Immuno-suppressive Agents |
azathioprine |
Imuran |
|
cyclosporine |
Neoral |
|
6-mercaptopurine |
Purinethol |
|
methotrexate |
|
|
Tumour Necrosis Factor-Alfa (TNF-alfa) Antagonists |
infliximab |
Remicade |
|
Corticosteroids |
|
|
|
Oral
|
budesonide |
Entocort capsule |
|
prednisone |
|
|
Rectal
|
betamethasone |
Betnesol enema |
|
budesonide |
Entocort enema |
|
hydrocortisone |
Cortenema, Cortifoam |
|
5-Aminosalicylic Acid Derivatives |
|
|
|
Oral
|
5-ASA (mesalamine) |
Asacol, Mesasal, Pentasa, Salofalk |
|
olsalazine |
Dipentum |
|
sulfasalazine |
Salazopyrin |
|
Rectal
|
5-ASA (mesalamine) |
Pentasa, Salofalk |
|
sulfasalazine |
Salazopyrin |
|
Drug Class |
Generic Name(s) |
Trade Name(s) |
|
|
|
|
|
Antiperistaltic opioid derivatives |
codeine phosphate |
|
|
diphenoxylate |
Lomotil |
|
loperamide |
Imodium |
|
Adsorbents
|
attapulgite |
Kaopectate |
|
cholestyramine |
Questran |
|
polycarbophil calcium |
Equalactin, Prodiem Bulk Fibre Therapy Caplets |
|
Antisecretory Agents |
octreotide |
Sandostatin |
|
Bismuth Compounds |
bismuth subsalicylate (+/- calcium carbonate) |
Pepto-Bismol |
|
Bulk-forming
|
methylcellulose |
Prodiem Bulk Fibre Therapy Powder |
|
psyllium |
Metamucil |
|
Probiotics |
Lactobacillus species |
Bacid |
|
Saccharomyces boulardii |
Florastar |
Antiflatulents |
simethicone |
Gas-X, Ovol, Phazyme |
Somatostatin Analogues |
octreotide |
Sandostatin |
|
somatostatin |
Stilamin |
|
Antinauseants and Antiemetic Agents |
|
|
|
Antihistamines |
dimenhydrinate |
Gravol |
|
diphenhydramine |
Benadryl |
|
doxylamine + pyridoxine |
Diclectin |
|
hydroxyzine |
Atarax |
|
meclizine |
Bonamine |
|
promethazine |
|
|
Anticholinergic Agents |
scopolamine |
Transderm V |
|
Dopamine Antagonists |
droperidol |
|
|
metoclopramide |
|
|
perphenazine |
Trilafon |
|
prochlorperazine |
Stemetil |
|
Serotonin (5-HT3) Antagonists |
dolasetron |
Anzemet |
|
granisetron |
Kytril |
|
ondansetron |
Zofran |
|
Drug Class |
Generic Name(s) |
Trade Name(s) |
|
Antinauseants and Antiemetic Agents |
|
|
|
Corticosteroids |
dexamethasone |
Dexasone |
|
methylprednisolone |
Medrol, Solu Medrol |
|
Benzodiazepines |
lorazepam |
Ativan |
|
Cannabinoids |
dronabinol |
Marinol |
|
nabilone |
Cesamet |
|
|
|