Gastrointestinal System – Drugs

(Products approved for use in Canada)

Drug Class

Generic Name(s)

Trade Name(s)

Antacids

aluminum hydroxide

Amphojel

aluminum hydroxide + magnesium hydroxide

Diovol, Gelusil, Maalox

calcium carbonate

Tums

calcium carbonate + magnesium hydroxide

Rolaids

magnesium hydroxide

Phillips' Milk of Magnesia

Antacid + Mucosal Anesthetic

oxethazaine + aluminum and magnesium hydroxide

Mucaine

Alginate + Antacid

alginic acid + aluminum hydroxide

Gaviscon

Prokinetic Agents

domperidone

erythromycin

EES, Erybid, Eryc, Erythrocin

metoclopramide

H2 receptor Antagonists

cimetidine

famotidine

Pepcid, Pepcid AC

nizatidine

Axid

ranitidine

Zantac

Proton-Pump Inhibitors

esomeprazole

Nexium

lansoprazole

Prevacid

omeprazole

Losec

pantoprazole

Pantoloc, Panto IV

rabeprazole

Pariet

Digestants (pancreatic enzymes)

pancrelipase

Cotazym, Creon, Pancrease, Ultrase, Viokase

Litholytic Agents (gallstone dissolution)

ursodeoxycholic acid or ursodiol

Urso

Drug Class

Generic Name(s)

Trade Name(s)

Antiviral Agents for Chronic Hepatitis

interferon alfa-2a

Roferon-A

interferon alfa-2b

Intron A

interferon alfacon-1

Infergen

lamivudine

Heptovir

peginterferon alfa-2a

Pegasys

peginterferon alfa-2b

Unitron PEG

ribavirin + interferon alfa-2a

Pegasys RBV

ribavirin + interferon alfa-2b

Rebetron

ribavirin + peginterferon alfa-2b

Pegetron

Hepatitis Vaccines

hepatitis A vaccine (inactivated)

Avaxim, Epaxal, Havrix, Vaqta

hepatitis B vaccine (recombinant)

Energix-B, Recombivax HB

hepatitis A & B vaccine

Twinrix

Cytoprotective Agents

misoprostol

sucralfate

Sulcrate

Laxatives

Bulk-forming agents

methylcellulose

Prodiem Bulk Fibre Therapy Powder

polycarbophil calcium

Prodiem Bulk Fibre Therapy Caplets

psyllium

Metamucil, Prodiem

sterculia gum

Normacol

Stimulants

bisacodyl

Carters Little Pills, Correctol, Dulcolax, Feen-A-Mint,

cascara sagrada

castor oil

senna

Ex-Lax, Nature’s Remedy, Prodiem Overnight Relief Therapy, Senokot

Stool softeners

docusate calcium or sodium

Colace, Correctol Stool Softener

Osmotic laxatives

glycerin

Suppositories

lactulose

polyethylene glycol (PEG) + electrolytes

Colyte, Klean-Prep, Lyteprep, PegLyte

sorbitol

Drug Class

Generic Name(s)

Trade Name(s)

Laxatives

Saline

magnesium citrate

Citro-Mag

magnesium hydroxide

Phillips Milk of Magnesia

sodium phosphates

Fleet Enema, Fleet Phosphosoda Oral Laxative,

Lubricants

mineral oil

Fleet Enema Mineral Oil, Lansoyl, Nujol,

Antispasmodics

Anticholinergics

dicyclomine

Bentylol

glycopyrrolate

hyoscine butylbromide

Buscopan

propantheline

Propanthel

Immuno-suppressive Agents

azathioprine

Imuran

cyclosporine

Neoral

6-mercaptopurine

Purinethol

methotrexate

Tumour Necrosis Factor-Alfa (TNF-alfa) Antagonists

infliximab

Remicade

Corticosteroids

Oral

budesonide

Entocort capsule

prednisone

Rectal

betamethasone

Betnesol enema

budesonide

Entocort enema

hydrocortisone

Cortenema, Cortifoam

5-Aminosalicylic Acid Derivatives

Oral

5-ASA (mesalamine)

Asacol, Mesasal, Pentasa, Salofalk

olsalazine

Dipentum

sulfasalazine

Salazopyrin

Rectal

5-ASA (mesalamine)

Pentasa, Salofalk

sulfasalazine

Salazopyrin

Drug Class

Generic Name(s)

Trade Name(s)

 

Antiperistaltic opioid derivatives

codeine phosphate

diphenoxylate

Lomotil

loperamide

Imodium

Adsorbents

attapulgite

Kaopectate

cholestyramine

Questran

polycarbophil calcium

Equalactin, Prodiem Bulk Fibre Therapy Caplets

Antisecretory Agents

octreotide

Sandostatin

Bismuth Compounds

bismuth subsalicylate (+/- calcium carbonate)

Pepto-Bismol

Bulk-forming

methylcellulose

Prodiem Bulk Fibre Therapy Powder

psyllium

Metamucil

Probiotics

Lactobacillus species

Bacid

Saccharomyces boulardii

Florastar

Antiflatulents

simethicone

Gas-X, Ovol, Phazyme

Somatostatin Analogues

octreotide

Sandostatin

somatostatin

Stilamin

Antinauseants and Antiemetic Agents

Antihistamines

dimenhydrinate

Gravol

diphenhydramine

Benadryl

doxylamine + pyridoxine

Diclectin

hydroxyzine

Atarax

meclizine

Bonamine

promethazine

Anticholinergic Agents

scopolamine

Transderm V

Dopamine Antagonists

droperidol

metoclopramide

perphenazine

Trilafon

prochlorperazine

Stemetil

Serotonin (5-HT3) Antagonists

dolasetron

Anzemet

granisetron

Kytril

ondansetron

Zofran

Drug Class

Generic Name(s)

 Trade Name(s)

Antinauseants and Antiemetic Agents

Corticosteroids

dexamethasone

Dexasone

methylprednisolone

Medrol, Solu Medrol

Benzodiazepines

lorazepam

Ativan

Cannabinoids

dronabinol

Marinol

nabilone

Cesamet






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